Browsing by Author Pandit, Amit

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Showing results 1 to 8 of 8
Issue DateTitleAuthor(s)
2021-04-30Design, synthesis and biological evaluation of enzyme inhibitorsChelvam, Venkatesh; Pandit, Amit
2025Design, synthesis, and biological evaluation of novel thiourea derivatives as small molecule inhibitors for prostate specific membrane antigenSengupta, Sagnik; Pandit, Amit; Krishnan, Mena Asha; Chelvam, Venkatesh
2025Design, Synthesis, and Cytotoxic Evaluation of New Structurally Simplified and Highly Potent Third-Generation Tubulysin DerivativesYadav, Kratika; Sharma, Lekhnath; Pandit, Amit; Pathak, Biswarup; Dräger, Gerald; Kirschning, Andreas; Venkatesh, Chelvam
2018First report on 3D-QSAR and molecular dynamics based docking studies of GCPII inhibitors for targeted drug delivery applicationsPandit, Amit; Sengupta, Sagnik; Krishnan, Mena Asha; Reddy, Ramesh B.; Chelvam, Venkatesh
2022Imaging of prostate cancer: optimizing affinity to prostate specific membrane antigen by spacer modifications in a tumor spheroid modelKrishnan, Mena Asha; Pandit, Amit; Chelvam, Venkatesh
2018In Vivo Evaluation of Ligand Targeted Drug Conjugates for Cancer TherapyKrishnan, Mena Asha; Pandit, Amit; Chelvam, Venkatesh
2021Structure activity relationships (SAR) study to design and synthesize new tubulin inhibitors with enhanced anti-tubulin activity: In silico and in vitro analysisPandit, Amit; Yadav, Kratika; Reddy, Ramesh B.; Sengupta, Sagnik; Chelvam, Venkatesh
2019Tyrosine-based asymmetric urea ligand for prostate carcinoma: Tuning biological efficacy through in silico studiesSengupta, Sagnik; Krishnan, Mena Asha; Pandit, Amit; Dudhe, Premansh; Chelvam, Venkatesh